Skelaxin (metaxalone) imagwiritsidwa ntchito pofuna kupweteka kwa minofu ndi kuuma kwachisokonezo chomwe chimakhudza kwambiri, zovuta za minofu monga kupweteka, kupopera, kapena kuvulala kwina. Nthawi zambiri amagwiritsidwa ntchito pophatikizapo mpumulo, mankhwala opatsirana.
Mapulogalamuwa amaperekedwa monga 5 - [(3,5- (dimethylphenoxy) methyl] -2-oxazolidinone ndi mawonekedwe a C12H15N03 ndi maselo olemera a 221.25.
Mankhwalawa samadziwika bwino, koma akatswiri amakhulupirira kuti mankhwalawa amagwira ntchito poletsa kusokonezeka kwa mitsempha kapena kupweteka mu ubongo.
Skelaxin imapezeka ndi mankhwala okhaokha ndipo ingaperekedwe kwa odwala omwe ali ndi zifukwa zotsatirazi:
- Kuthamanga kwa minofu
- Chidwi mu Cerebral palsy
- Kumva kupweteka kumbuyo kapena kupweteka kwa mutu
- Fibromyalgia
- Kuthetsa mutu kumutu
- Matenda a myofascial syndrome
- Multiple sclerosis
Ndondomeko Yoperekedwa
Mlingo wotchuka wa Skelaxin kwa akuluakulu ndi ana oposa zaka 12 ndi piritsi imodzi ya 800 mg katatu kapena kanayi patsiku. Ndikofunika kuti musamamwe mankhwala ambiri kuposa dokotala wanu. Zotsatira zoopsa zingachitike ngati mutenga zambiri.
Skelaxin imalowa m'matumbo aang'ono ndipo imayambitsidwa ndi chiwindi komanso imatulutsa mkodzo ngati ma metabolites osadziwika.
Amene sayenera kutenga Skelaxin
Ngakhale kuti Skelaxin yapezeka kuti ili otetezeka kwa odwala ambiri, odwala ena sayenera kuwatenga.
Izi zikuphatikizapo odwala aliwonse omwe amadziwika kuti hypersensitivity kwa zigawo zilizonse za mankhwala; omwe ali ndi chizolowezi chodziwika ndi mankhwala osokoneza bongo, hemolytic, kapena anemias; ndi omwe ali ndi vuto lalikulu kwambiri la chibwibwi kapena kugwira ntchito.
Kuonjezera apo, odwala omwe amamwa mowa ayenera kulangizidwa kuti Skelaxin ikhoze kukweza zotsatira za mowa ndi zina za CNS zosautsa.
Zingasokoneze malingaliro aumunthu ndi / kapena thupi kuti athe kuchita ntchito zoopsa, monga kugwiritsa ntchito makina kapena kuyendetsa galimoto, makamaka ngati akugwiritsidwa ntchito mowa kapena ena oponderezedwa ndi CNS.
Kugwiritsidwa ntchito mosasamala kwa metaxalone sikungakhazikitsidwe pokhudzana ndi zomwe zingawononge zotsatira za kukula kwa mwana. Choncho, mapiritsi a Skelaxin sayenera kugwiritsidwa ntchito kwa amayi omwe ali ndi pakati kapena makamaka omwe ali ndi pakati pomwe pokhapokha ngati wodwalayo ali ndi mwayi wopambana pangozi zoopsa.
Sikudziwika ngati mankhwalawa amavutsidwira mkaka waumunthu. Monga lamulo, asamwino sayenera kuchitidwa pamene wodwala ali ndi mankhwala chifukwa mankhwala ambiri amawotcha mkaka waumunthu. Kugwiritsidwa ntchito kwa ana, chitetezo ndi mphamvu kwa ana a zaka khumi ndi ziwiri ndi pansi sizinakhazikitsidwe .
Zotsatira Zotsatira
Ngakhale kuti ndizosawerengeka, zotsatira za anaphylactoid zafotokozedwa ndi Skelaxin. Zizindikilo zowonongeka zikuphatikizapo:
- Mikoko
- Kuvuta kupuma
- Kutupa kwa nkhope, milomo, lilime, kapena mmero
- Kugona ndi chizungulire
- Nausea
- Kuthamanga
Kuchita kawirikawiri kwa metaxalone ndi:
- CNS: kugona, chizungulire, kupweteka mutu, ndi mantha kapena "kukwiya"
- Kudwala: kunyoza, kusanza, kukwiya kwa m'mimba
- Chitetezo chautetezo: Kuthamanga kwa thupi kumatulutsa, kuthamanga kapena popanda pruritus
- Hematologic: leukopenia, hemolytic anemia
- Hepatobiliary: jaundice
> Chitsime:
US Food and Drug Administration, NDA 13-217 / S-036, Revised: August, 2002