Methimazole / Tapazole kwa Matenda a Manda

Matenda a Antithyroid Akugwira Ntchito Yopereka Matenda a Manda ndi Hyperthyroidism

Mankhwala a Antithyroid - amatchedwanso thioamides - ndi mankhwala omwe amachititsa chithokomiro choopsa (hyperthyroidism) mwa kuteteza khungu la chithokomiro kuti lichititse mahomoni a chithokomiro. Pochizira chithokomiro chochulukirapo, chomwe chimachokera ku matenda omwe amadziwika ndi dzina lakuti Graves 'matenda, ndizofunika kuchepetsa kuchulukitsa kwa mavitamini a chithokomiro, makamaka mahomoni thyroxine (T4) ndi triiodothyronine (T3).

Mankhwala a Antithyroid amachititsa kuti zikhale zovuta kwambiri kuti thupi lizigwiritsa ntchito ayodini, motero amaletsa mapangidwe a mahomoni a chithokomiro.

Thandizo la mankhwala a Antithyroid ndi limodzi mwa mankhwala okhudzana ndi hyperthyroidism ndi matenda a Graves. Njira zina zothandizira mankhwalawa zimaphatikizapo kupuma kwa ayodini (RAI) ndi kupititsa patsogolo mankhwala onse kapena mbali ina ya chithokomiro .

Pali mankhwala awiri ofunikira omwe alipo tsopano ku United States: propylthiouracil (PTU) ndi methimazole. Ku United States, methimazole imatengedwa kuti ndi mankhwala osakaniza antithyroid nthawi zambiri.

Methimazole, nthawi zina amatchedwa thiamazole, amaletsa chithokomiro kuti asagwiritse ntchito ayodini kuti apange mahomoni a chithokomiro. Nthawi zambiri amatengedwa ngati mlingo kamodzi patsiku.

Mankhwalawa amagwiritsidwa ntchito kuzungulira dziko lapansi. Ku United States, Tapazole ndi dzina lokha la mankhwala otchedwa antithyroid mankhwala a methimazole. Pali opanga ojambula ambiri a methimazole.

Tapazole

Tapazole ndi dzina la methimazole , mankhwala osokoneza bongo omwe amapangidwa ndi King Pharmaceuticals, Inc. The FDA inavomereza Tapazole mu 2000.

Zosakaniza Tapazole : methimazole USP; lactose monohydrate; magnesium stearate; chomera (chimanga); chomera chosakaniza; ndi talc.

Mphamvu Zilipo : 5 mg ndi 10 mg

Generic Methimazole (ndi Sandoz)

Sandoz, membala wa Novartis Group of Companies, amapanga methimazole yachibadwa. Inavomerezedwa ndi FDA mu 2001.

Sandoz Methimazole Zosakaniza: methimazole USP; lactose monohydrate; magnesium stearate; chomera (chimanga); ndi talc.

Mphamvu Zilipo: 5 mg ndi 10 mg

Generic Methimazole (ndi Cedar Pharmaceuticals LLC)

Cedar Pharmaceuticals LLC amapanga methimazole omwe amaperekedwa ndi United Research Laboratories. Chivomerezo cha FDA chinapezeka mu 2005.

Cedar Pharmaceuticals Methimazole Zosakaniza: methimazole USP; chodabwitsa; magnesium stearate; wowuma wa mbatata; ndi talc.

Mphamvu Zilipo: 5 mg, 10 mg, 15 mg, 20 mg

Generic Methimazole (mwa Activis Totowa)

Activis Totowa LLC opanga methimazole generic ndi FDA adalandira mu 2007.

Activis Methimazole Zosakaniza methimazole USP; lactose monohydrate; magnesium stearate; starch pregelatinized; ndi talc.

Mphamvu zilipo: 5 mg ndi 10 mg

Generic Methimazole (mwa Caraco Pharmaceutical Laboratories)

Caraco Pharmaceutical Laboratories, Ltd. ikupanga methimazole yomwe inavomerezedwa ndi FDA mu 2007.

Caraco Methimazole Zosakaniza: methimazole USP; lactose monohydrate; povidone; talc; chithunzi; magnesium stearate; ndi wowuma chimanga.

Mphamvu Zilipo : 5mg ndi 10mg

Generic Methimazole (mwa Par Pharmaceutical Companies)

Par Pharmaceutical Companies amapanga methimazole yowonjezera.

Zosakaniza: methimazole USP; lactose monohydrate; magnesium stearate; chimanga cha chimanga; ndi talc.

Mphamvu Zilipo: 5 mg ndi 10 mg

Zotsatira:

Daily Med, US Chakudya Chakumwa Chakumwa Chakumwa kwa Mankhwala.

Kulankhulana Kwachidakwa kwa FDA: Kuchenjezedwa Kwatsopano kwa Chiwindi Choopsa Ndi Propylthiouracil, pa 21 April 2010

Ross, Douglas MD, "Wodwala mankhwala: mankhwala osokoneza bongo," UpToDate . Idasinthidwa komaliza: November 13, 2009

Malipoti owonjezera ndi: Leslie Blumenberg